Cloning, Characterization, and Sulfonamide and Thiol Inhibition Studies of an α-Carbonic Anhydrase from Trypanosoma cruzi, the Causative Agent of Chagas Disease

Author:

Pan Peiwen1,Vermelho Alane Beatriz2,Capaci Rodrigues Giseli2,Scozzafava Andrea3,Tolvanen Martti E. E.1,Parkkila Seppo1,Capasso Clemente4,Supuran Claudiu T.35

Affiliation:

1. Institute of Biomedical Technology, Fimlab Ltd., School of Medicine and BioMediTech, University of Tampere and Tampere University Hospital, Medisiinarinkatu 3, 33520 Tampere, Finland

2. Laboratório Proteases de Microrganismos, Instituto de Microbiologia Paulo de Góes, Universidade Federal do Rio de Janeiro, UFRJ, CCS, Bloco I, Sala 32, Cidade Universitária, Av. Carlos Chagas Filho, 373, Ilha do Fundão, Rio de Janeiro R.J., Brazil

3. Laboratorio di Chimica Bioinorganica, Rm. 188, Polo Scientifico, Università degli Studi di Firenze, Via della Lastruccia 3, 50019 Sesto Fiorentino, Florence, Italy

4. Istituto di Biochimica delle Proteine, CNR, Via P. Castellino 111, 80131 Napoli, Italy

5. Dipartimento di Scienze Farmaceutiche, Università degli Studi di Firenze, Via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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