Spectral and Crystallographic Study of Pyridinic Analogues of Nimesulide: Determination of the Active Form of Methanesulfonamides as COX-2 Selective Inhibitors-Reference-Cited by-同舟云学术

Spectral and Crystallographic Study of Pyridinic Analogues of Nimesulide: Determination of the Active Form of Methanesulfonamides as COX-2 Selective Inhibitors

Published:2002-10-03 Issue:23 Volume:45 Page:5182-5185
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Julémont Fabien¹,de Leval Xavier¹,Michaux Catherine¹,Damas Jacques¹,Charlier Caroline¹,Durant François¹,Pirotte Bernard¹,Dogné Jean-Michel¹

Affiliation:

1. Natural and Synthetic Drugs Research Center, Department of Medicinal Chemistry, Université de Liège, 1, Avenue de l'Hôpital, Tour 4(+5) Sart-Tilman, B-4000 Liège, Belgium, Department of Molecular and Structural Chemistry, Université de Namur, 61 Rue de Bruxelles, B-5000 Namur, Belgium, and Department of Human Physiology, Université de Liège, 17 Place Delcour, 4020 Liège, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020920n

Reference13 articles.

1. Cyclooxygenase inhibitors – current status and future prospects

2. Constitutive cyclooxygenase (COX-1) and inducible cyclooxygenase (COX-2): Rationale for selective inhibition and progress to date

Cited by 34 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Isonimesulide and Its Carborane Analogues as Isoform‐Selective COX Inhibitors and Antitumor Agents;Advanced Therapeutics;2023-05-24

2. Nimesulide analogues: From anti-inflammatory to antitumor agents;Bioorganic Chemistry;2019-07

3. Triazolopyrimidine and triazolopyridine scaffolds as TDP2 inhibitors;Bioorganic & Medicinal Chemistry Letters;2019-01

4. Atom-based QSAR and 3D QSAR using pharmacophore based alignment for discovery of nimesulide-derived SKBR-3 cell line inhibitors;Medicinal Chemistry Research;2014-07-31

5. Time-Dependent Diaryl Ether Inhibitors of InhA: Structure-Activity Relationship Studies of Enzyme Inhibition, Antibacterial Activity, and in vivo Efficacy;ChemMedChem;2014-03-11