Thecis-4-Amino-l-proline Residue as a Scaffold for the Synthesis of Cyclic and Linear Endomorphin-2 Analogues-Reference-Cited by-同舟云学术

Thecis-4-Amino-l-proline Residue as a Scaffold for the Synthesis of Cyclic and Linear Endomorphin-2 Analogues

Published:2012-03-22 Issue:7 Volume:55 Page:3027-3035
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mollica Adriano¹,Pinnen Francesco¹,Stefanucci Azzurra¹,Feliciani Federica¹,Campestre Cristina¹,Mannina Luisa²³,Sobolev Anatoly P.³,Lucente Gino⁴,Davis Peg,Lai Josephine,Ma Shou-Wu,Porreca Frank,Hruby Victor J.

Affiliation:

1. Dipartimento di Scienze del Farmaco, Università di Chieti-Pescara “G. d’Annunzio”, Via dei Vestini 31, 66100 Chieti, Italy

2. Dipartimento di Chimica e Tecnologie del Farmaco, “La Sapienza” Università di Roma, P.le A. Moro 5, 00185 Rome, Italy

3. Istituto di Metodologie Chimiche, Laboratorio di Risonanza Magnetica “Annalaura Segre”, CNR, Via Salaria Km 29.300, 00015 Monterotondo, Rome, Italy

4. Dipartimento di Chimica e Tecnologie del Farmaco e Istituto di Chimica Biomolecolare, CNR Sezione di Roma, “La Sapienza” Università di Roma, P.le A. Moro 5, 00185 Roma, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201402v

Reference46 articles.

1. A potent and selective endogenous agonist for the µ-opiate receptor

2. Synthesis and evaluation of new endomorphin analogues modified at the Pro2 residue

3. Synthesis and Evaluation of New Endomorphin-2 Analogues Containing (Z)-α,β-Didehydrophenylalanine (ΔZPhe) Residues

4. Synthesis and activity of endomorphin-2 and morphiceptin analogues with proline surrogates in position 2

5. Peptides and the blood-brain barrier

Cited by 33 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis, characterization, and biological study of new synthetic opioid hemorphin‐4 peptides containing sterically restricted nonnatural amino acids;Archiv der Pharmazie;2024-04-05

2. Evaluation of Antimicrobial Activities against Various E. coli Strains of a Novel Hybrid Peptide—LENART01;Molecules;2023-06-23

3. Harnessing the cyclization strategy for new drug discovery;Acta Pharmaceutica Sinica B;2022-12

4. Selective MOR activity of DAPEA and Endomorphin-2 analogues containing a (R)-γ-Freidinger lactam in position two;Bioorganic Chemistry;2021-10

5. An Effective and Safe Enkephalin Analog for Antinociception;Pharmaceutics;2021-06-22