Bis-Quinolinium Cyclophanes: 6,10-Diaza-3(1,3),8(1,4)-dibenzena-1,5(1,4)- diquinolinacyclodecaphane (UCL 1684), the First Nanomolar, Non-Peptidic Blocker of the Apamin-Sensitive Ca2+-Activated K+ Channel-Reference-Cited by-同舟云学术

Bis-Quinolinium Cyclophanes: 6,10-Diaza-3(1,3),8(1,4)-dibenzena-1,5(1,4)- diquinolinacyclodecaphane (UCL 1684), the First Nanomolar, Non-Peptidic Blocker of the Apamin-Sensitive Ca2+-Activated K+ Channel

Published:1998-01-01 Issue:1 Volume:41 Page:2-5
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rosa Joaquin Campos¹,Galanakis Dimitrios¹,Ganellin C. Robin¹,Dunn Philip M.¹,Jenkinson Donald H.¹

Affiliation:

1. Departments of Chemistry and Pharmacology, University College London, Gower Street, London WC1E 6BT, U.K., Departamento de Quimica Organica, Facultad de Farmacia, Universidad de Granada, Campus de Cartuja, s/n, 18071 Granada, Spain, and Department of Pharmaceutical Chemistry, School of Pharmacy, Aristotelian University of Thessaloniki, Thessaloniki, 540 06, Greece

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970571a

Reference39 articles.

1. (a) Haylett, D. G.; Jenkinson, D. H. InPotassium Channels; Cook, N. S., Ed.; Ellis Horwood Limited: Chichester, 1990; pp 70−95.

2. Expression of apamin receptor in muscles of patients with myotonic muscular dystrophy

3. Increase of apamin receptors in skeletal muscle induced by colchicine: possible role in myotonia

4. Possible role of apamin-sensitive K+ channels in myotonic dystrophy

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