1-[2-Methoxy-5-(3-phenylpropyl)]-2-aminopropane Unexpectedly Shows 5-HT2A Serotonin Receptor Affinity and Antagonist Character-Reference-Cited by-同舟云学术

1-[2-Methoxy-5-(3-phenylpropyl)]-2-aminopropane Unexpectedly Shows 5-HT2A Serotonin Receptor Affinity and Antagonist Character

Published:2001-08-30 Issue:20 Volume:44 Page:3283-3291
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rangisetty Jagadeesh B.¹,Dukat Małgorzata¹,Dowd Cynthia S.¹,Herrick-Davis Katharine¹,DuPre Ann¹,Gadepalli Sami¹,Teitler Milt¹,Kelley Curtis R.¹,Sharif Najam A.¹,Glennon Richard A.¹

Affiliation:

1. Department of Medicinal Chemistry, School of Pharmacy, Virginia Commonwealth University, Richmond, Virginia 23298-0540, Center for Neuropharmacology and Neuroscience, Albany Medical College, Albany, New York 12208, and Alcon Laboratories Inc., 6201 South Freeway, Fort Worth, Texas 76134-2099

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0100739

Reference25 articles.

1. Van Wijngaarden, I.; Soudijn, W. 5-HT2A, 5-HT2B, and 5-HT2Creceptor ligands. InSerotonin Receptors and their Ligands; Olivier, B., van Wijngaarden, I., Soudijn, W., Eds.; Elsevier: Amsterdam, 1997; pp 161−197.

2. A structure-affinity study of the binding of 4-substituted analogs of 1-(2,5-dimethoxyphenyl)-2-aminopropane at 5-HT2 serotonin receptors

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