Development of the Commercial Route for the Manufacture of a 5-Lipoxygenase Inhibitor PF-04191834-Reference-Cited by-同舟云学术

Development of the Commercial Route for the Manufacture of a 5-Lipoxygenase Inhibitor PF-04191834

Published:2015-12-11 Issue:12 Volume:19 Page:1944-1953
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Chekal Brian¹,Damon David¹,LaFrance Danny¹,Leeman Kyle¹,Mojica Carlos¹,Palm Andrew¹,St. Pierre Michael¹,Sieser Janice¹,Sutherland Karen¹,Vaidyanathan Rajappa¹,Van Alsten John¹,Vanderplas Brian¹,Wager Carrie¹,Weisenburger Gerald¹,Withbroe Gregory¹,Yu Shu¹

Affiliation:

1. Chemical Research and Development, Pfizer Worldwide R&D-Groton Laboratories, 558 Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op500412a

Reference41 articles.

1. Alvira, E.; Graneto, M. J.; Grapperhaus, M. L.; Iyanar, K.; Maddux, T. M.; Mahoney, M. W.; Massa, M. A.; Sample, R. K.; Schmidt, M. A.; Seidel, R. E.; Selbo, J. G.; Tollefson, M. B.; Vonder Embse, R. A.; Wagner, G. M.; Woodard, S. S.WO 2009069044 A1, 2009.

2. Graneto, M. J.; Maddux, T. M.; Masferrer, J. L.US 20080125474 A1, 2008.

3. Development an Efficient Route to the 5-Lipoxygenase Inhibitor PF-04191834

4. Optimization of Imidazole 5-Lipoxygenase Inhibitors and Selection and Synthesis of a Development Candidate

5. 5-Lipoxygenase inhibitors: convenient synthesis of 4-[3-(4-heterocyclylphenylthio)phenyl]-3,4,5,6-tetrahydro-2H-pyran-4-carboxamide analogues

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