Extensive Rigid Analogue Design Maps the Binding Conformation of Potent N-Benzylphenethylamine 5-HT2A Serotonin Receptor Agonist Ligands-Reference-Cited by-同舟云学术

Extensive Rigid Analogue Design Maps the Binding Conformation of Potent N-Benzylphenethylamine 5-HT2A Serotonin Receptor Agonist Ligands

Published:2012-08-01 Issue:1 Volume:4 Page:96-109
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Juncosa Jose I.¹,Hansen Martin¹,Bonner Lisa A.¹,Cueva Juan Pablo¹,Maglathlin Rebecca¹,McCorvy John D.¹,Marona-Lewicka Danuta¹,Lill Markus A.¹,Nichols David E.¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, West Lafayette, Indiana 47907, United States

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/cn3000668

Reference26 articles.

1. Serotonin Receptors

2. Siegel, G. J. and Agranoff, B. W. (1999) Basic neurochemistry: molecular, cellular, and medical aspects,6th ed., pxxi,1183,Lippincott-Raven Publishers,Philadelphia.

3. Serotonin receptor modulation in irritable bowel syndrome: one step forwards and one step backwards

4. Role of the Serotonin 5-HT2A Receptor in Learning

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