Synthesis and Evaluation of Estrogen Receptor Ligands with Bridged Oxabicyclic Cores Containing a Diarylethylene Motif: Estrogen Antagonists of Unusual Structure-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Estrogen Receptor Ligands with Bridged Oxabicyclic Cores Containing a Diarylethylene Motif: Estrogen Antagonists of Unusual Structure

Published:2005-10-18 Issue:23 Volume:48 Page:7261-7274
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhou Hai-Bing¹,Comninos John S.¹,Stossi Fabio¹,Katzenellenbogen Benita S.¹,Katzenellenbogen John A.¹

Affiliation:

1. Department of Chemistry and Department of Molecular and Integrative Physiology, University of Illinois, 600 South Mathews Avenue, Urbana, Illinois 61801

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0506773

Reference41 articles.

1. ERβ: Identification and characterization of a novel human estrogen receptor

2. Cloning of a novel receptor expressed in rat prostate and ovary.

3. Comparative distribution of estrogen receptor-? and -? mRNA in the rat central nervous system

4. Comparative distribution of estrogen receptor-α (ER-α) and β (ER-β) mRNA in the rat pituitary, gonad, and reproductive tract

5. Tissue Distribution and Quantitative Analysis of Estrogen Receptor-α (ERα) and Estrogen Receptor-β (ERβ) Messenger Ribonucleic Acid in the Wild-Type and ERα-Knockout Mouse

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