Nicotinamide Phosphoribosyltransferase Inhibitors, Design, Preparation, and Structure–Activity Relationship

Author:

Christensen Mette K.1,Erichsen Kamille D.1,Olesen Uffe H.12,Tjørnelund Jette1,Fristrup Peter3,Thougaard Annemette1,Nielsen Søren Jensby1,Sehested Maxwell12,Jensen Peter B.1,Loza Einars4,Kalvinsh Ivars4,Garten Antje5,Kiess Wieland5,Björkling Fredrik16

Affiliation:

1. Topotarget A/S, Symbion, Fruebjergvej 3, Copenhagen DK-2100, Denmark

2. Experimental Pathology Unit, National University Hospital, Biocentre, Ole Maaloes Vej 5, Copenhagen DK-2200, Denmark

3. Department of Chemistry, Technical University of Denmark, Kemitorvet 207, Lyngby DK-2800, Denmark

4. Latvian Institute of Organic Synthesis, Aizkraukles 21, Riga LV-1006, Latvia

5. Center for Pediatric Research, Hospital for Children and Adolescents, University of Leipzig, Liebigstr. 21, Leipzig 04301, Germany

6. Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, Copenhagen DK-2100, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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