Discovery of Novel Benzoxaborole-Based Potent Antitrypanosomal Agents

Author:

Ding Dazhong1,Zhao Yaxue1,Meng Qingqing1,Xie Dongsheng1,Nare Bakela2,Chen Daitao2,Bacchi Cyrus J.3,Yarlett Nigel3,Zhang Yong-Kang4,Hernandez Vincent4,Xia Yi4,Freund Yvonne4,Abdulla Maha5,Ang Kean-Hooi5,Ratnam Joseline5,McKerrow James H.5,Jacobs Robert T.2,Zhou Huchen1,Plattner Jacob J.4

Affiliation:

1. School of Pharmacy and E-Institute of Chemical Biology, Shanghai Jiao Tong University, Shanghai, 200240, China

2. SCYNEXIS, Inc., P.O. Box 12878, Research Triangle Park, North Carolina 27709

3. Haskins Laboratory, Pace University, New York, New York 10038

4. Anacor Pharmaceuticals Inc., 1020 East Meadow Circle, Palo Alto, California 94303

5. Small Molecule Discovery Center and Sandler Center for Basic Research in Parasitic Diseases, University of California, San Francisco, California 94158

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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