In Vitro and in Vivo Evaluation of 6-Azido-2‘,3‘-dideoxy-2‘-fluoro-β-d-arabinofuranosylpurine and N6-Methyl-2‘,3‘-dideoxy-2‘-fluoro-β-d-arabinofuranosyladenine as Prodrugs of the Anti-HIV Nucleosides 2‘-F-ara-ddA and 2‘-F-ara-ddI-Reference-Cited by-同舟云学术

In Vitro and in Vivo Evaluation of 6-Azido-2‘,3‘-dideoxy-2‘-fluoro-β-d-arabinofuranosylpurine and N6-Methyl-2‘,3‘-dideoxy-2‘-fluoro-β-d-arabinofuranosyladenine as Prodrugs of the Anti-HIV Nucleosides 2‘-F-ara-ddA and 2‘-F-ara-ddI

Published:1996-01-01 Issue:23 Volume:39 Page:4676-4681
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Koudriakova Tanya¹,Manouilov Konstantine K.¹,Shanmuganathan Kirupa¹,Kotra Lakshmi P.¹,Boudinot F. Douglas¹,Cretton-Scott Erica¹,Sommadossi Jean-Pierre¹,Schinazi Raymond F.¹,Chu Chung K.¹

Affiliation:

1. Departments of Medicinal Chemistry and Pharmaceutics, College of Pharmacy, The University of Georgia, Athens, Georgia 30602-2352, Department of Pharmacology, School of Medicine, University of Alabama, Birmingham, Alabama 35294, and Veterans Affairs Medical Center and Department of Pediatrics, Emory University School of Medicine, Atlanta, Georgia 30033

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960140c

Reference16 articles.

1. Impact of bioavailability on determination of the maximal tolerated dose of 2',3'-dideoxyinosine in phase I trials

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