Deconstruction of the α4β2 Nicotinic Acetylcholine Receptor Positive Allosteric Modulator Desformylflustrabromine
Author:
Affiliation:
1. Department of Medicinal Chemistry, School of Pharmacy, Virginia Commonwealth University, Richmond, Virginia 23298, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm200834x
Reference17 articles.
1. Nicotinic Acetylcholine Receptors and Nicotinic Cholinergic Mechanisms of the Central Nervous System
2. Molecular mechanisms and binding site locations for noncompetitive antagonists of nicotinic acetylcholine receptors
3. Positive and negative modulation of nicotinic receptors
4. Allosteric modulation of nicotinic acetylcholine receptors
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2. Synthesis of β-Carbolines with Electrocyclic Cyclization of 3-Nitrovinylindoles;International Journal of Molecular Sciences;2023-08-23
3. Desformylflustrabromine (dFBr), a positive allosteric modulator of the α4β2 nicotinic receptor modulates the hypnotic response to ethanol;Alcohol;2021-06
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