Discovery of Ligands for ADP-Ribosyltransferases via Docking-Based Virtual Screening-Reference-Cited by-同舟云学术

Discovery of Ligands for ADP-Ribosyltransferases via Docking-Based Virtual Screening

Published:2012-08-20 Issue:17 Volume:55 Page:7706-7718
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Andersson C. David¹,Karlberg Tobias²,Ekblad Torun²,Lindgren Anders E. G.¹,Thorsell Ann-Gerd²,Spjut Sara¹,Uciechowska Urszula¹,Niemiec Moritz S.¹,Wittung-Stafshede Pernilla¹,Weigelt Johan²,Elofsson Mikael¹,Schüler Herwig²,Linusson Anna¹

Affiliation:

1. Department of Chemistry, Umeå University, SE-90187 Umeå, Sweden

2. Department of Medical Biochemistry and Biophysics, Karolinska Institutet, SE-17177 Stockholm, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300746d

Reference69 articles.

1. Toward a unified nomenclature for mammalian ADP-ribosyltransferases

2. The diverse biological roles of mammalian PARPS, a small but powerful family of poly-ADP-ribose polymerases

3. A review of PARP inhibitors: from bench to bedside

4. B-aggressive Lymphoma Family Proteins Have Unique Domains That Modulate Transcription and Exhibit Poly(ADP-ribose) Polymerase Activity

5. Substrate-Assisted Catalysis by PARP10 Limits Its Activity to Mono-ADP-Ribosylation

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