Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt, d-2-Nal4]endomorphin-1 (Antanal-1) and [Dmt1, d-2-Nal4]endomorphin-2 (Antanal-2)-Reference-Cited by-同舟云学术

Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt, d-2-Nal4]endomorphin-1 (Antanal-1) and [Dmt1, d-2-Nal4]endomorphin-2 (Antanal-2)

Published:2007-01-09 Issue:3 Volume:50 Page:512-520
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fichna Jakub¹,do-Rego Jean-Claude¹,Chung Nga N.¹,Lemieux Carole¹,Schiller Peter W.¹,Poels Jeroen¹,Vanden Broeck Jozef¹,Costentin Jean¹,Janecka Anna¹

Affiliation:

1. Laboratory of Biomolecular Chemistry, Institute of Biomedicinal Chemistry, Medical University, Lodz, Poland, Laboratoire de Neuropsychopharmacologie Expérimentale, CNRS-FRE 2735, IFRMP 23, Université de Rouen, France, Laboratory of Chemical Biology and Peptide Research, Clinical Research Institute of Montreal, Montreal, Canada, and Laboratory for Developmental Physiology, Genomics and Proteomics, Zoological Institute, Catholic University, Leuven, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060998u

Reference35 articles.

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4. Binaltorphimine and nor-binaltorphimine, potent and selective k-opioid receptor antagonists

5. TIPP[.psi.]: a highly potent and stable pseudopeptide .delta. opioid receptor antagonist with extraordinary .delta. selectivity

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