From Poor Substrates to Good Inhibitors: Design of Inhibitors for Serine and Thiol Proteases
Author:
Affiliation:
1. Brandeis University, 415 South Street, Waltham, Massachusetts 02254
Publisher
American Chemical Society (ACS)
Subject
Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/bi952879e
Reference11 articles.
1. Fersht, A. (1984)Enzyme Structure & Mechanism, 2nd ed., p 317, W. H. Freeman & Co., New York.
2. Aromatic esters which inhibit plasmin or thrombin by formation of relatively stable acyl enzymes
3. Cysteine protease inhibition by azapeptide esters
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