A Novel Palladium-Mediated Coupling Approach to 2,3-Disubstituted Benzo[b]thiophenes and Its Application to the Synthesis of Tubulin Binding Agents-Reference-Cited by-同舟云学术

A Novel Palladium-Mediated Coupling Approach to 2,3-Disubstituted Benzo[b]thiophenes and Its Application to the Synthesis of Tubulin Binding Agents

Published:2001-02-06 Issue:5 Volume:3 Page:651-654
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Flynn Bernard L.¹,Verdier-Pinard Pascal¹,Hamel Ernest¹

Affiliation:

1. Department of Chemistry, The Faculties, Australian National University, Canberra, ACT, 0200, Australia, and Screening Technologies Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, National Cancer Institute, Frederick Cancer Research and Development Center, Frederick, Maryland 21702

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ol0067179

Reference34 articles.

1. Recent Advances in the Synthesis and Applications of Benzo[b]thiophenes

2. Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-[2-(1-piperidinyl)ethoxy]phenyl]methanone hydrochloride (LY 156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity

3. Selective Estrogen Receptor Modulators: An Alternative to Hormone Replacement Therapy

4. A new anti-tubulin agent containing the benzo[b]thiophene ring system

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