Discovery of 3-Substituted Aminocyclopentanes as Potent and Orally Bioavailable NR2B Subtype-Selective NMDA Antagonists-Reference-Cited by-同舟云学术

Discovery of 3-Substituted Aminocyclopentanes as Potent and Orally Bioavailable NR2B Subtype-Selective NMDA Antagonists

Published:2011-06-20 Issue:7 Volume:2 Page:352-362
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Layton Mark E.¹,Kelly Michael J.¹,Rodzinak Kevin J.¹,Sanderson Philip E.¹,Young Steven D.¹,Bednar Rodney A.¹,DiLella Anthony G.¹,Mcdonald Terrence P.¹,Wang Hao¹,Mosser Scott D.¹,Fay John F.¹,Cunningham Michael E.¹,Reiss Duane R.¹,Fandozzi Christine¹,Trainor Nicole¹,Liang Annie¹,Lis Edward V.¹,Seabrook Guy R.¹,Urban Mark O.¹,Yergey James¹,Koblan Kenneth S.¹

Affiliation:

1. Departments of †Medicinal Chemistry, ‡Molecular Pain Research, §Movement Disorders, and ∥Drug Metabolism, Merck Research Laboratories, West Point, Pennsylvania 19486, United States

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/cn200013d

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