6β-Acyloxy(nor)tropanes: Affinities for Antagonist/Agonist Binding Sites on Transfected and Native Muscarinic Receptors
Author:
Affiliation:
1. Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm9904001
Reference28 articles.
1. Selective Muscarinic Receptor Agonists and Antagonists
2. Muscarinic Receptors—Characterization, coupling and function
3. Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo-M ratio as an index of efficacy at cortical muscarinic receptors
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1. Medicinal chemistry and therapeutic potential of muscarinic M3 antagonists;Medicinal Research Reviews;2009-11
2. Quantitative determination of a novel enantiomeric tropane analog, (−)-satropane, in biological fluids using liquid chromatography/tandem mass spectrometry;Biomedical Chromatography;2009-10
3. Docking analyses on human muscarinic receptors: Unveiling the subtypes peculiarities in agonists binding;Bioorganic & Medicinal Chemistry;2008-03-15
4. Stereoselectivity of satropane, a novel tropane analog, on iris muscarinic receptor activation and intraocular hypotension;Acta Pharmacologica Sinica;2008-02
5. Novel oxotremorine-related heterocyclic derivatives: Synthesis and in vitro pharmacology at the muscarinic receptor subtypes;Bioorganic & Medicinal Chemistry;2007-12
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