Converting Potent Indeno[1,2-b]indole Inhibitors of Protein Kinase CK2 into Selective Inhibitors of the Breast Cancer Resistance Protein ABCG2-Reference-Cited by-同舟云学术

Converting Potent Indeno[1,2-b]indole Inhibitors of Protein Kinase CK2 into Selective Inhibitors of the Breast Cancer Resistance Protein ABCG2

Published:2014-10-16 Issue:1 Volume:58 Page:265-277
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Jabor Gozzi Gustavo¹²,Bouaziz Zouhair³,Winter Evelyn¹⁴,Daflon-Yunes Nathalia¹,Aichele Dagmar⁵,Nacereddine Abdelhamid³,Marminon Christelle³,Valdameri Glaucio¹²,Zeinyeh Waël³,Bollacke Andre⁵,Guillon Jean⁶,Lacoudre Aline⁷,Pinaud Noël⁷,Cadena Silvia M.²,Jose Joachim⁵,Le Borgne Marc³,Di Pietro Attilio¹

Affiliation:

1. Equipe Labellisée Ligue 2014, BMSSI UMR 5086 CNRS/Université Lyon 1, IBCP, 69367 Lyon, France

2. Department of Biochemistry and Molecular Biology, Federal University of Paraná, Curitiba, Paraná 80060-000, Brazil

3. Université de Lyon, Université Lyon 1, Faculté de Pharmacie, ISPB, EA 4446 Biomolécules Cancer et Chimiorésistances, SFR Santé Lyon-Est CNRS UMS3453-INSERM US7, 8 Avenue Rockefeller, F-69373 Lyon Cedex 8, France

4. Department of Pharmaceutical Sciences, PGFAR, Federal University of Santa Catarina, Florianopolis, Santa Catarina 88040-900, Brazil

5. Institute of Pharmaceutical and Medicinal Chemistry, PharmaCampus, Westfälische Wilhelms-University Münster, Corrensstrasse 48, 48149 Münster, Germany

6. Université de Bordeaux, UFR des Sciences Pharmaceutiques, INSERM U869, Laboratoire ARNA, 146 Rue Léo Saignat, F-33076 Bordeaux Cedex, France

7. ISM-CNRS UMR 5255, Université de Bordeaux, 351 Cours de la Libération, F-33405 Talence Cedex, France

Funder

Agence Nationale de la Recherche

Conselho Nacional de Desenvolvimento Científico e Tecnológico

Ligue Contre le Cancer

Coordenação de Aperfeiçoamento de Pessoal de Nível Superior

Nemzeti Innovációs Hivatal

Centre National de la Recherche Scientifique

Publisher

American Chemical Society (ACS)

Subject