Benzothiazepinone Binding Domain of Purified L-Type Calcium Channels: Direct Labeling Using a Novel Fluorescent Diltiazem Analog-Reference-Cited by-同舟云学术

Benzothiazepinone Binding Domain of Purified L-Type Calcium Channels: Direct Labeling Using a Novel Fluorescent Diltiazem Analog

Published:1995-03 Issue:10 Volume:34 Page:3461-3469
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Brauns Thomas,Cai Zhen-Wei,Kimball S. David,Kang Hee-Chol,Haugland Richard P.,Berger Wolfgang,Berjukov Stanislav,Hering Steffen,Glossmann Hartmut,Striessnig Joerg

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi00010a039

Reference28 articles.

1. Complex Molecular Mechanism for Dihydropyridine Binding to L-Type Ca2+-Channels As Revealed by Fluorescence Resonance Energy Transfer

2. Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

3. Purification of a functional receptor for calcium-channel blockers from rabbit skeletal-muscle microsomes

4. Benzazepinone calcium channel blockers. 2. Structure activity and drug metabolism studies leading to potent antihypertensive agents. Comparison with benzothiazepinones

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5. Molecular Mechanism of Diltiazem Interaction with L-type Ca2+ Channels;Journal of Biological Chemistry;1998-10