Synthesis, Anti-Inflammatory Activity, and in Vitro Antitumor Effect of a Novel Class of Cyclooxygenase Inhibitors: 4-(Aryloyl)phenyl Methyl Sulfones-Reference-Cited by-同舟云学术

Synthesis, Anti-Inflammatory Activity, and in Vitro Antitumor Effect of a Novel Class of Cyclooxygenase Inhibitors: 4-(Aryloyl)phenyl Methyl Sulfones

Published:2010-08-30 Issue:18 Volume:53 Page:6560-6571
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Harrak Youssef¹,Casula Giovanni²,Basset Joan¹,Rosell Glòria¹,Plescia Salvatore²,Raffa Demetrio²,Cusimano Maria Grazia²,Pouplana Ramon³,Pujol Maria Dolors¹

Affiliation:

1. Laboratori de Química Farmacèutica (Unitat Associada al CSIC)

2. Dipartamento di Chimica e Tecnologie Farmaceutiche, Facoltà di Farmacia, Università degli Studi di Palermo, Via Archirafi, 32-90123 Palermo, Italy

3. Laboratori de Físico-Química

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100398z

Reference45 articles.

1. Selective COX-2 Inhibitors and Dual Acting Anti-inflammatory Drugs: Critical Remarks

2. Synthesis and biological evaluation of N-difluoromethyl-1,2-dihydropyrid-2-one acetic acid regioisomers: Dual Inhibitors of cyclooxygenases and 5-lipoxygenase

3. Synthesis of Celecoxib Analogues Possessing a N-Difluoromethyl-1,2-dihydropyrid-2-one 5-Lipoxygenase Pharmacophore: Biological Evaluation as Dual Inhibitors of Cyclooxygenases and 5-Lipoxygenase with Anti-Inflammatory Activity

4. Cyclooxygenase inhibitors – current status and future prospects

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