Discovery and Optimization of Sulfonyl Acrylonitriles as Selective, Covalent Inhibitors of Protein Phosphatase Methylesterase-1-Reference-Cited by-同舟云学术

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Discovery and Optimization of Sulfonyl Acrylonitriles as Selective, Covalent Inhibitors of Protein Phosphatase Methylesterase-1

Published:2011-07-28 Issue:14 Volume:54 Page:5229-5236
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bachovchin Daniel A.,Zuhl Andrea M.,Speers Anna E.,Wolfe Monique R.,Weerapana Eranthie,Brown Steven J.,Rosen Hugh,Cravatt Benjamin F.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200502u

Reference39 articles.

1. Serine/Threonine Phosphatases: Mechanism through Structure

2. Regulation of protein kinase cascades by protein phosphatase 2A

3. Regulation of Protein Serine-Threonine Phosphatase Type-2A by Tyrosine Phosphorylation

4. Autophosphorylation-activated protein kinase phosphorylates and inactivates protein phosphatase 2A.

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