Mechanism of Inhibition of the GluA2 AMPA Receptor Channel Opening: The Role of 4-Methyl versus 4-Carbonyl Group on the Diazepine Ring of 2,3-Benzodiazepine Derivatives
Author:
Affiliation:
1. Department of Chemistry, and Center for Neuroscience Research, University at Albany, SUNY, Albany, New York 12222, United States
2. Dipartimento Farmaco-Chimico, Università di Messina, viale Annunziata, 98168 Messina, Italy
Publisher
American Chemical Society (ACS)
Subject
Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/cn200033j
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1. The Molecular Pharmacology and Cell Biology of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid Receptors
2. Quinoxalinediones: Potent Competitive Non-NMDA Glutamate Receptor Antagonists
3. ZK200775: A phosphonate quinoxalinedione AMPA antagonist for neuroprotection in stroke and trauma
4. synthesis and Structure-Activity Relationships of 2,3-Benzodiazepines as AMPA Receptor Antagonists
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