Dual RXR Agonists and RAR Antagonists Based on the Stilbene Retinoid Scaffold-Reference-Cited by-同舟云学术

Dual RXR Agonists and RAR Antagonists Based on the Stilbene Retinoid Scaffold

Published:2014-03-21 Issue:5 Volume:5 Page:533-537
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Martínez Claudio¹,Lieb Michele²,Álvarez Susana¹,Rodríguez-Barrios Fátima¹,Álvarez Rosana¹,Khanwalkar Harshal²,Gronemeyer Hinrich²,de Lera Angel R.¹

Affiliation:

1. Departamento de Química Orgánica, Facultade de Química, CINBIO, Universidade de Vigo, and Instituto de Investigación Biomédica de Vigo (IBIV), 36310 Vigo, Spain

2. Equipe Labellisée Ligue Contre le Cancer, Department of Functional Genomics and Cancer, Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)/CNRS/INSERM/UdS, BP 10142, 67404 Illkirch, Cedex, C. U. de Strasbourg, France

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml400521f

Reference47 articles.

1. Visualization of an endogenous retinoic acid gradient across embryonic development

2. FUNCTION OF RETINOID NUCLEAR RECEPTORS: Lessons from Genetic and Pharmacological Dissections of the Retinoic Acid Signaling Pathway During Mouse Embryogenesis

3. RAR and RXR modulation in cancer and metabolic disease

4. Retinoic acid in development: towards an integrated view

5. International Union of Pharmacology. LX. Retinoic Acid Receptors

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