Active-Site Inhibitors Modulate the Dynamic Properties of Human Monoacylglycerol Lipase: A Hydrogen Exchange Mass Spectrometry Study-Reference-Cited by-同舟云学术

Active-Site Inhibitors Modulate the Dynamic Properties of Human Monoacylglycerol Lipase: A Hydrogen Exchange Mass Spectrometry Study

Published:2013-07-08 Issue:29 Volume:52 Page:5016-5026
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Karageorgos Ioannis¹,Wales Thomas E.²,Janero David R.¹,Zvonok Nikolai¹,Vemuri V. Kiran¹,Engen John R.²,Makriyannis Alexandros¹

Affiliation:

1. Center for Drug Discovery and Departments of Pharmaceutical Sciences and Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115-5000, United States

2. Department of Chemistry and Chemical Biology and Barnett Institute of Chemical and Biological Analysis, Northeastern University, Boston, Massachusetts 02115-5000, United States

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi400430k

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4. Biosynthesis and degradation of the endocannabinoid 2-arachidonoylglycerol

5. The pharmacological landscape and therapeutic potential of serine hydrolases

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