A New Class of Nonpeptide Bradykinin B2 Receptor Ligand, Incorporating a 4-Aminoquinoline Framework. Identification of a Key Pharmacophore To Determine Species Difference and Agonist/Antagonist Profile-Reference-Cited by-同舟云学术

A New Class of Nonpeptide Bradykinin B2 Receptor Ligand, Incorporating a 4-Aminoquinoline Framework. Identification of a Key Pharmacophore To Determine Species Difference and Agonist/Antagonist Profile

Published:2004-04-01 Issue:10 Volume:47 Page:2667-2677
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sawada Yuki¹,Kayakiri Hiroshi¹,Abe Yoshito¹,Mizutani Tsuyoshi¹,Inamura Noriaki¹,Asano Masayuki¹,Aramori Ichiro¹,Hatori Chie¹,Oku Teruo¹,Tanaka Hirokazu¹

Affiliation:

1. Exploratory Research Laboratories, Fujisawa Pharmaceutical Co. Ltd., 5-2-3 Tokodai, Tsukuba, Ibaraki 300-2698, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030326t

Reference38 articles.

1. Neuron atrophy during aging: programmed or sporadic?

2. Expression cloning of a rat B2 bradykinin receptor.

3. Potent, long-acting bradykinin antagonists for a wide range of applications

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