Regioselective Suzuki Coupling of Dihaloheteroaromatic Compounds as a Rapid Strategy To Synthesize Potent Rigid Combretastatin Analogues-Reference-Cited by-同舟云学术

Regioselective Suzuki Coupling of Dihaloheteroaromatic Compounds as a Rapid Strategy To Synthesize Potent Rigid Combretastatin Analogues

Published:2011-07-28 Issue:14 Volume:54 Page:4977-4986
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Theeramunkong Sewan,Caldarelli Antonio,Massarotti Alberto,Aprile Silvio,Caprioglio Diego,Zaninetti Roberta,Teruggi Alessia,Pirali Tracey,Grosa Giorgio,Tron Gian Cesare,Genazzani Armando A.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm200555r

Reference32 articles.

1. Isolation and structure of the strong cell growth and tubulin inhibitor combretastatin A-4

2. Combretastatin anticancer drugs

3. The tumor vascular targeting agent combretastatin A–4-phosphate induces reorganization of the actin cytoskeleton and early membrane blebbing in human endothelial cells

4. The development of combretastatin A4 phosphate as a vascular targeting agent

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