Receptor-Based Pharmacophores for Serotonin 5-HT7R AntagonistsImplications to Selectivity-Reference-Cited by-同舟云学术

Receptor-Based Pharmacophores for Serotonin 5-HT7R AntagonistsImplications to Selectivity

Published:2006-10-20 Issue:23 Volume:49 Page:6732-6741
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kołaczkowski Marcin¹,Nowak Mateusz¹,Pawłowski Maciej¹,Bojarski Andrzej J.¹

Affiliation:

1. Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, 12 Smȩtna Street, 31-343 Kraków, Poland, and Department of Pharmaceutical Chemistry, Collegium Medicum, Jagiellonian University, 9 Medyczna Street, 30-688 Kraków, Poland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060300c

Reference65 articles.

1. Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation.

2. A novel adenylyl cyclase-activating serotonin receptor (5-HT7) implicated in the regulation of mammalian circadian rhythms

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