Evolution of the Thienopyridine Class of Inhibitors of IκB Kinase-β: Part I: Hit-to-Lead Strategies-Reference-Cited by-同舟云学术

Evolution of the Thienopyridine Class of Inhibitors of IκB Kinase-β: Part I: Hit-to-Lead Strategies

Published:2006-04-20 Issue:10 Volume:49 Page:2898-2908
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Morwick Tina¹,Berry Angela¹,Brickwood Janice¹,Cardozo Mario¹,Catron Katrina¹,DeTuri Molly¹,Emeigh Jonathan¹,Homon Carol¹,Hrapchak Matt¹,Jacober Stephen¹,Jakes Scott¹,Kaplita Paul¹,Kelly Terence A.¹,Ksiazek John¹,Liuzzi Michel¹,Magolda Ronald¹,Mao Can¹,Marshall Daniel¹,McNeil Daniel¹,Prokopowicz Anthony¹,Sarko Christopher¹,Scouten Erika¹,Sledziona Cynthia¹,Sun Sanxing¹,Watrous Jane¹,Wu Jiang Ping¹,Cywin Charles L.¹

Affiliation:

1. Boehringer Ingelheim Pharmaceuticals, Inc., 900 Ridgebury Road, Ridgefield, Connecticut 06801-0368, and Boehringer Ingelheim (Canada) Ltd., 2100 Cunard Street, Laval (Quebec), Canada H7S 2G5

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0510979

Reference42 articles.

1. Components of Successful Lead Generation

2. Lead Generation - Enhancing the Success of Drug Discovery by Investing in the Hit to Lead Process

3. Lead Generation: Sowing the Seeds for Future Success

4. Drugs, leads, and drug-likeness: an analysis of some recently launched drugs

Cited by 68 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Fused Pyridine Derivatives: Synthesis and Biological Activities;Exploring Chemistry with Pyridine Derivatives;2023-01-04

2. Recent developments in oxidative functionalization reactions promoted by TBAI/TBHP;Synthetic Communications;2021-12-02

3. Synthesis of Biologically Active Heterocycles via a Domino Sequence Involving an SN2/Thorpe–Ziegler Reaction Step;Synthesis;2021-06-10

4. 2-Cyclopropyl-6-phenyl-2,3-dihydrothieno[3,2-d][1,3,2]diazaborinin-4(1H)-one;Molbank;2021-06-01

5. Synthesis and characterization of 1,2,4-triazolo[1,5-a]pyrimidine-2-carboxamide-based compounds targeting the PA-PB1 interface of influenza A virus polymerase;European Journal of Medicinal Chemistry;2021-01