Using Fragment Cocktail Crystallography To Assist Inhibitor Design of Trypanosoma brucei Nucleoside 2-Deoxyribosyltransferase-Reference-Cited by-同舟云学术

Using Fragment Cocktail Crystallography To Assist Inhibitor Design of Trypanosoma brucei Nucleoside 2-Deoxyribosyltransferase

Published:2006-09-02 Issue:20 Volume:49 Page:5939-5946
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bosch Jürgen¹,Robien Mark A.¹,Mehlin Christopher¹,Boni Erica¹,Riechers Aaron¹,Buckner Frederick S.¹,Van Voorhis Wesley C.¹,Myler Peter J.¹,Worthey Elizabeth A.¹,DeTitta George¹,Luft Joseph R.¹,Lauricella Angela¹,Gulde Stacey¹,Anderson Lori A.¹,Kalyuzhniy Oleksandr¹,Neely Helen M.¹,Ross Jenni¹,Earnest Thomas N.¹,Soltis Michael¹,Schoenfeld Lori¹,Zucker Frank¹,Merritt Ethan A.¹,Fan Erkang¹,Verlinde Christophe L. M. J.¹,Hol Wim G. J.¹

Affiliation:

1. Department of Biochemistry, Division of Infectious Disease, and Howard Hughes Medical Institute, University of Washington, Seattle, Washington 98195, Structural Genomics of Pathogenic Protozoa (SGPP) Consortium, Seattle, Washington 98185, Seattle Biomedical Research Institute, Seattle, Washington 98109, Hauptmann-Woodward Institute, Buffalo, New York 14203, Physical Biosciences Division, Lawrence Berkeley National Laboratory, Berkeley, California 94720, and SSRL, Stanford University, Stanford, California...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060429m

Reference34 articles.

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