Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion-Reference-Cited by-同舟云学术

Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion

Published:2010-02-12 Issue:5 Volume:53 Page:2038-2050
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Carmi Caterina¹,Cavazzoni Andrea²,Vezzosi Stefano¹,Bordi Fabrizio¹,Vacondio Federica¹,Silva Claudia¹,Rivara Silvia¹,Lodola Alessio¹,Alfieri Roberta R.²,La Monica Silvia²,Galetti Maricla²,Ardizzoni Andrea³,Petronini Pier Giorgio²,Mor Marco¹

Affiliation:

1. Dipartimento Farmaceutico, Università degli Studi di Parma, V.le G.P. Usberti 27/A, I-43124 Parma, Italy

2. Dipartimento di Medicina Sperimentale, Università degli Studi di Parma, Via Volturno 39, I-43125 Parma, Italy

3. Oncologia Medica, Azienda Ospedaliero—Universitaria di Parma, V.le Gramsci 14, I-43126 Parma, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm901558p

Reference67 articles.

1. Untangling the ErbB signalling network

2. Epidermal Growth Factor Receptor Copy Number Alterations Correlate With Poor Clinical Outcome in Patients With Head and Neck Squamous Cancer

3. Studies leading to the identification of ZD1839 (iressa™): an orally active, selective epidermal growth factor receptor tyrosine kinase inhibitor targeted to the treatment of cancer

4. Activating Mutations in the Epidermal Growth Factor Receptor Underlying Responsiveness of Non–Small-Cell Lung Cancer to Gefitinib

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