Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)-Reference-Cited by-同舟云学术

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

Published:1999-03-01 Issue:6 Volume:42 Page:1053-1065
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Giardina Giuseppe A. M.¹,Raveglia Luca F.¹,Grugni Mario¹,Sarau Henry M.¹,Farina Carlo¹,Medhurst Andrew D.¹,Graziani Davide¹,Schmidt Dulcie B.¹,Rigolio Roberto¹,Luttmann Mark¹,Cavagnera Stefano¹,Foley James J.¹,Vecchietti Vittorio¹,Hay Douglas W. P.¹

Affiliation:

1. Department of Medicinal Chemistry, SmithKline Beecham S.p.A., Via Zambeletti, 20021 Baranzate, Milano, Italy, Department of Pulmonary Pharmacology, SmithKline Beecham Pharmaceuticals, 709 Swedeland Road, King of Prussia, Pennsylvania 19406-0939, and Department of Neurology Research, SmithKline Beecham Pharmaceuticals, New Frontiers Science Park, Third Avenue, Harlow, Essex, England CM19 5AW

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980633c

Reference37 articles.

1. Tachykinin receptors and tachykinin receptor antagonists

2. Tachykinins

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