Indolylarylsulfones Carrying a Heterocyclic Tail as Very Potent and Broad Spectrum HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors-Reference-Cited by-同舟云学术

Indolylarylsulfones Carrying a Heterocyclic Tail as Very Potent and Broad Spectrum HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors

Published:2014-11-24 Issue:23 Volume:57 Page:9945-9957
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Famiglini Valeria¹,La Regina Giuseppe¹,Coluccia Antonio¹,Pelliccia Sveva²,Brancale Andrea³,Maga Giovanni⁴,Crespan Emmanuele⁴,Badia Roger⁵,Riveira-Muñoz Eva⁵,Esté José A.⁵,Ferretti Rosella⁶,Cirilli Roberto⁶,Zamperini Claudio⁷,Botta Maurizio⁷,Schols Dominique⁸,Limongelli Vittorio²,Agostino Bruno²,Novellino Ettore²,Silvestri Romano¹

Affiliation:

1. Istituto Pasteur − Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, Piazzale Aldo Moro 5, I-00185 Roma, Italy

2. Dipartimento di Farmacia, Università di Napoli Federico II, Via Domenico Montesano 49, I-80131 Napoli, Italy

3. Welsh School of Pharmacy, Cardiff University, King Edward VII Avenue, Cardiff CF10 3NB, United Kingdom

4. Institute of Molecular Genetics IGM-CNR, National Research Council, via Abbiategrasso 207, I-27100 Pavia, Italy

5. AIDS Research Institute − IrsiCaixa, Hospitals Germans Trias i Pujol, Universitat Autonóma de Barcelona, 08916 Badalona, Spain

6. Dipartimento del Farmaco, Istituto Superiore di Sanità, Viale Regina Elena 299, I-00161 Roma, Italy

7. Dipartimento di Biotecnologia Chimica e Farmacia, Università di Siena, Via Aldo Moro 2, I-53100 Siena, Italy

8. Department of Microbiology and Immunology, University of Leuven, Minderbroedersstraat 10, 3000 Leuven, Belgium

Funder

KU Leuven

Ministerio de Economía y Competitividad

Fonds Wetenschappelijk Onderzoek

Istituto Pasteur-Fondazione Cenci Bolognetti

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5011622

Reference43 articles.

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