Distinguishing between the Permeability Relationships with Absorption and Metabolism To Improve BCS and BDDCS Predictions in Early Drug Discovery
Author:
Affiliation:
1. Department of Bioengineering and Therapeutic Sciences, University of California—San Francisco, San Francisco, California 94143-0912, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Pharmaceutical Science,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/mp4007858
Reference46 articles.
1. Screening for human ADME/Tox drug properties in drug discovery
2. Intestinal permeability and its relevance for absorption and elimination
3. Caco-2 replace or refine?
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