Identification of Cinnamic Acid Derivatives As Novel Antagonists of the Prokaryotic Proton-Gated Ion Channel GLIC-Reference-Cited by-同舟云学术

Identification of Cinnamic Acid Derivatives As Novel Antagonists of the Prokaryotic Proton-Gated Ion Channel GLIC

Published:2013-06-04 Issue:11 Volume:56 Page:4619-4630
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Prevost Marie S.¹²³,Delarue-Cochin Sandrine⁴⁵,Marteaux Justine⁴⁵,Colas Claire⁶⁷,Van Renterghem Catherine¹²,Blondel Arnaud⁶⁷,Malliavin Thérèse⁶⁷,Corringer Pierre-Jean¹²,Joseph Delphine⁴⁵

Affiliation:

1. Institut Pasteur, Unité Récepteurs-Canaux, Paris, France

2. CNRS UMR 3571, Paris, France

3. Université Pierre et Marie Curie (UPMC), Cellule Pasteur, Paris, France

4. Université Paris-Sud, Équipe de Chimie des Substances Naturelles, Châtenay-Malabry, France

5. CNRS UMR 8076 BioCIS, Châtenay-Malabry, France

6. Institut Pasteur, Unité de Bioinformatique Structurale, Paris, France

7. CNRS UMR 3528, Paris, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400374q

Reference47 articles.

1. Structure and Pharmacology of Pentameric Receptor Channels: From Bacteria to Brain

2. Principles of activation and permeation in an anion-selective Cys-loop receptor

3. Ligand Activation of the Prokaryotic Pentameric Ligand-Gated Ion Channel ELIC

4. Structure of the pentameric ligand-gated ion channel ELIC cocrystallized with its competitive antagonist acetylcholine

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