Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase-Reference-Cited by-同舟云学术

Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase

Published:2014-04-11 Issue:8 Volume:57 Page:3223-3234
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Costi Roberta¹,Métifiot Mathieu²,Chung Suhman³,Cuzzucoli Crucitti Giuliana¹,Maddali Kasthuraiah²,Pescatori Luca¹,Messore Antonella¹,Madia Valentina Noemi¹,Pupo Giovanni¹,Scipione Luigi¹,Tortorella Silvano¹,Di Leva Francesco Saverio⁴,Cosconati Sandro⁵,Marinelli Luciana⁴,Novellino Ettore⁴,Le Grice Stuart F. J.³,Corona Angela⁶,Pommier Yves²,Marchand Christophe²,Di Santo Roberto¹

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Istituto Pasteur-Fondazione Cenci Bolognetti, “Sapienza” Università di Roma, P.le Aldo Moro 5, I-00185 Roma, Italy

2. Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, 37 Convent Drive, Bethesda, Maryland 20892, United States

3. RT Biochemistry Section, HIV Drug Resistance Program, National Cancer Institute, Frederick, Maryland 21702, United States

4. Dipartimento di Farmacia, Università di Napoli “Federico II” Via D. Montesano 49, 80131 Napoli, Italy

5. DiSTABiF, Seconda Università di Napoli, Via Vivaldi 43, 81100 Caserta, Italy

6. Department of Life and Environmental Sciences, University of Cagliari, 09124 Cagliari, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm5001503

Reference80 articles.

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