Elesclomol-Copper Nanoparticles Overcome Multidrug Resistance in Cancer Cells
Author:
Affiliation:
1. Department of Drug Discovery and Development, Harrison College of Pharmacy, Auburn University, Auburn, Alabama 36849, United States
2. National Institute on Drug Abuse, 11601 Landsdown Street, North Bethesda, Maryland 20852, United States
Funder
Auburn University
Publisher
American Chemical Society (ACS)
Link
https://pubs.acs.org/doi/pdf/10.1021/acsami.3c17792
Reference54 articles.
1. Elesclomol: a copper ionophore targeting mitochondrial metabolism for cancer therapy
2. Elesclomol elevates cellular and mitochondrial iron levels by delivering copper to the iron import machinery
3. Mitochondrial metabolism promotes adaptation to proteotoxic stress
4. Copper induces cell death by targeting lipoylated TCA cycle proteins
5. Ferredoxin 1 is a cuproptosis-key gene responsible for tumor immunity and drug sensitivity: A pan-cancer analysis
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