Synthesis and Structure−Affinity−Activity Relationships of Novel Benzofuran Derivatives as MT2 Melatonin Receptor Selective Ligands-Reference-Cited by-同舟云学术

Synthesis and Structure−Affinity−Activity Relationships of Novel Benzofuran Derivatives as MT2 Melatonin Receptor Selective Ligands

Published:2002-05-18 Issue:13 Volume:45 Page:2788-2800
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wallez Valérie¹,Durieux-Poissonnier Sophie¹,Chavatte Philippe¹,Boutin Jean A.¹,Audinot Valérie¹,Nicolas Jean-Paul¹,Bennejean Caroline¹,Delagrange Philippe¹,Renard Pierre¹,Lesieur Daniel¹

Affiliation:

1. Institut de Chimie Pharmaceutique Albert Lespagnol, 3 rue du Professeur Laguesse, BP 83, 59006 Lille Cedex, France, Division de Pharmacologie Moléculaire et Cellulaire, Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France, and Institut de Recherches Internationales Servier, 1 rue Carle Hébert, 92415 Courbevoie Cedex, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0005252

Reference36 articles.

1. Pineal Melatonin: Cell Biology of Its Synthesis and of Its Physiological Interactions*

2. Molecular characterization of a second melatonin receptor expressed in human retina and brain: the Mel1b melatonin receptor.

3. Dubocovich, M.L.; Cardinali, D. P.; Delagrange, P.; Krause, D. N.; Strosberg, A. D.; Sugden, D.; Yocca, F. D.The IUPHAR Compendium ofReceptor Characterization and Classification; IUPHAR Media: London, 2000; pp 271−277.

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