Structure-Based Evaluation of Non-nucleoside Inhibitors with Improved Potency and Solubility That Target HIV Reverse Transcriptase Variants
Author:
Affiliation:
1. Department of Pharmacology, ‡Department of Chemistry, Yale University, New Haven, Connecticut 06520-8066, United States
Funder
National Institute of Allergy and Infectious Diseases
National Institute of General Medical Sciences
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm501908a
Reference35 articles.
1. Antiviral Drug Resistance and the Need for Development of New HIV-1 Reverse Transcriptase Inhibitors
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3. Anti-HIV drugs: 25 compounds approved within 25 years after the discovery of HIV
4. Rilpivirine: A second-generation nonnucleoside reverse transcriptase inhibitor
5. Treatment of HIV infection with once-daily regimens
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