N-Substituted cis-4a-(3-Hydroxyphenyl)-8a-methyloctahydroisoquinolines Are Opioid Receptor Pure Antagonists-Reference-Cited by-同舟云学术

N-Substituted cis-4a-(3-Hydroxyphenyl)-8a-methyloctahydroisoquinolines Are Opioid Receptor Pure Antagonists

Published:2005-11-16 Issue:26 Volume:48 Page:8182-8193
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Carroll F. Ivy¹,Chaudhari Sachin¹,Thomas James B.¹,Mascarella S. Wayne¹,Gigstad Kenneth M.¹,Deschamps Jeffrey¹,Navarro Hernán A.¹

Affiliation:

1. Organic and Medicinal Chemistry, Research Triangle Institute, Research Triangle Park, North Carolina 27709, and Laboratory for the Structure of Matter, Naval Research Laboratory, 4555 Overlook Avenue, Washington, D.C. 20375-5341

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm058261c

Reference30 articles.

1. 5′-Guanidinonaltrindole, a highly selective and potent κ-opioid receptor antagonist

2. Binaltorphimine and nor-binaltorphimine, potent and selective k-opioid receptor antagonists

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