Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor-Reference-Cited by-同舟云学术

Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor

Published:2004-10-05 Issue:6 Volume:48 Page:1813-1822
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Surleraux Dominique L. N. G.¹,Tahri Abdellah¹,Verschueren Wim G.¹,Pille Geert M. E.¹,de Kock Herman A.¹,Jonckers Tim H. M.¹,Peeters Anik¹,De Meyer Sandra¹,Azijn Hilde¹,Pauwels Rudi¹,de Bethune Marie-Pierre¹,King Nancy M.¹,Prabu-Jeyabalan Moses¹,Schiffer Celia A.¹,Wigerinck Piet B. T. P.¹

Affiliation:

1. Tibotec BVBA, Generaal de Wittelaan L 11B 3, B-2800 Mechelen, Belgium, and Department of Biochemistry and Molecular Pharmacology, University of Massachusetts Medical School, Worcester, Massachusetts 01605

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049560p

Reference28 articles.

1. Overview of the effectiveness of triple combination therapy in antiretroviral-naive HIV-1 infected adults

2. Declining Morbidity and Mortality among Patients with Advanced Human Immunodeficiency Virus Infection

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