Modified Cap Group Suberoylanilide Hydroxamic Acid Histone Deacetylase Inhibitor Derivatives Reveal Improved Selective Antileukemic Activity-Reference-Cited by-同舟云学术

Modified Cap Group Suberoylanilide Hydroxamic Acid Histone Deacetylase Inhibitor Derivatives Reveal Improved Selective Antileukemic Activity

Published:2010-03-10 Issue:8 Volume:53 Page:3038-3047
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Salmi-Smail Chanaz¹,Fabre Aurélie¹,Dequiedt Franck²,Restouin Audrey¹,Castellano Rémy¹,Garbit Slaveia¹,Roche Philippe³,Morelli Xavier³,Brunel Jean Michel⁴,Collette Yves¹

Affiliation:

1. Unité 891 INSERM, Centre de Recherche en Cancérologie de Marseille, 27 bd Lei Roure, 13009 Marseille 09, France

2. Cellular and Molecular Biology Unit, Fonds National de la Recherche Scientifique, Faculté Universitaire des Sciences Agronomiques de Gembloux, 13 Av. Maréchal Juin, B-5030 Gembloux, Belgium

3. CNRS-IBSM, IMR Laboratory, 31 Chemin de Joseph Aiguier, 13402 Marseille 20, France

4. Laboratoire URMITE UMR 6236 CNRS, Faculté de Médecine et de Pharmacie, Université de la Méditerranée, 27 bd Jean Moulin, 13385 Marseille 05, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm901358y

Reference39 articles.

1. Roles of histone acetyltransferases and deacetylases in gene regulation

2. Histone deacetylase inhibitors and the promise of epigenetic (and more) treatments for cancer

3. Regulating the Regulators

4. Histone Deacetylase Inhibition Selectively Alters the Activity and Expression of Cell Cycle Proteins Leading to Specific Chromatin Acetylation and Antiproliferative Effects

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