Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1-Reference-Cited by-同舟云学术

Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1

Published:2014-01-28 Issue:4 Volume:5 Page:422-427
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Fader Lee D.¹,Malenfant Eric¹,Parisien Mathieu¹,Carson Rebekah¹,Bilodeau François¹,Landry Serge¹,Pesant Marc¹,Brochu Christian¹,Morin Sébastien¹,Chabot Catherine¹,Halmos Ted¹,Bousquet Yves¹,Bailey Murray D.¹,Kawai Stephen H.¹,Coulombe René¹,LaPlante Steven¹,Jakalian Araz¹,Bhardwaj Punit K.¹,Wernic Dominik¹,Schroeder Patricia¹,Amad Ma’an¹,Edwards Paul¹,Garneau Michel¹,Duan Jianmin¹,Cordingley Michael¹,Bethell Richard¹,Mason Stephen W.¹,Bös Michael¹,Bonneau Pierre¹,Poupart Marc-André¹,Faucher Anne-Marie¹,Simoneau Bruno¹,Fenwick Craig¹,Yoakim Christiane¹,Tsantrizos Youla¹

Affiliation:

1. Research and Development, Boehringer Ingelheim (Canada) Ltd., 2100 Cunard Street, Laval, Québec H7S 2G5, Canada

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml500002n

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