Selection and Development of the Manufacturing Route for EP1 Antagonist GSK269984B
Author:
Affiliation:
1. Synthetic Chemistry, Chemical Development, GlaxoSmithKline, Gunnels Wood Road, Stevenage, Hertfordshire SG1 2NY, U.K.
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/op100072y
Reference49 articles.
1. Novel methylene-linked heterocyclic EP1 receptor antagonists
2. bGiblin, G. M. P.; Hall, A.; Hurst, D. N.; Scoccitti, T.PCT Int. Appl. WO 2007128752(CAN 147:541735), 2007.
3. Discovery of sodium 6-[(5-chloro-2-{[(4-chloro-2-fluorophenyl)methyl]oxy}phenyl)methyl]-2-pyridinecarboxylate (GSK269984A) an EP1 receptor antagonist for the treatment of inflammatory pain
4. Giblin, G. M. P.; Hall, A.; Hurst, D. N.; Rawlings, D. A.; Scoccitti, T.PCT Int. Appl. WO 2006066968(CAN 145:83231), 2006.
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