Synthesis and Evaluation of Aryl-Naloxamide Opiate Analgesics Targeting Truncated Exon 11-Associated μ Opioid Receptor (MOR-1) Splice Variants-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Aryl-Naloxamide Opiate Analgesics Targeting Truncated Exon 11-Associated μ Opioid Receptor (MOR-1) Splice Variants

Published:2012-07-16 Issue:14 Volume:55 Page:6352-6362
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Majumdar Susruta¹,Subrath Joan¹,Le Rouzic Valerie¹,Polikar Lisa¹,Burgman Maxim¹,Nagakura Kuni¹,Ocampo Julie¹,Haselton Nathan¹,Pasternak Anna R.¹,Grinnell Steven¹,Pan Ying-Xian¹,Pasternak Gavril W.¹

Affiliation:

1. Molecular Pharmacology and Chemistry Program and Department of Neurology, Memorial Sloan-Kettering Cancer Center, 1275 York Avenue, New York, New York 10065, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300305c

Reference43 articles.

1. Dissociation of morphine's analgesic and respiratory depressant actions

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