Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar-Reference-Cited by-同舟云学术

Potent and Selective Inhibitors of Breast Cancer Resistance Protein (ABCG2) Derived from the p-Glycoprotein (ABCB1) Modulator Tariquidar

Published:2009-01-26 Issue:4 Volume:52 Page:1190-1197
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kühnle Matthias¹,Egger Michael¹,Müller Christine¹,Mahringer Anne¹,Bernhardt Günther¹,Fricker Gert¹,König Burkhard¹,Buschauer Armin¹

Affiliation:

1. Department of Pharmaceutical/Medicinal Chemistry II, Institute of Pharmacy, and Institute of Organic Chemistry, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstrasse 31, D-93053 Regensburg, Germany, Institute of Pharmacy and Molecular Biotechnology, University of Heidelberg, Im Neuenheimer Feld 366, D-69120 Heidelberg, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm8013822

Reference44 articles.

1. Do cMOAT (MRP2), other MRP homologues, and LRP play a role in MDR?

2. The role of the human ABCG2 multidrug transporter and its variants in cancer therapy and toxicology

3. ABCG2: determining its relevance in clinical drug resistance

Cited by 143 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Development and validation of an LC-MS/MS method for simultaneous quantification of eight drugs in plasma and brain: Application in a pharmacokinetic study in mice;Journal of Chromatography B;2024-09

2. ATP-binding cassette transporter inhibitor potency and substrate drug affinity are critical determinants of successful drug delivery enhancement to the brain;Fluids and Barriers of the CNS;2024-08-05

3. Breast Cancer Resistance Protein: Structure, Localization, Functions, Significance for Rational Pharmacotherapy;I.P. Pavlov Russian Medical Biological Herald;2024-07-10

4. Strategies to enhance the response of liver cancer to pharmacological treatments;American Journal of Physiology-Cell Physiology;2024-07-01

5. Triazoles in Medicinal Chemistry: Physicochemical Properties, Bioisosterism, and Application;Journal of Medicinal Chemistry;2024-05-03