Human cytochromes P450 mediating phenacetin O‐deethylation in vitro: Validation of the high affinity component as an index of CYP1A2 activity-Reference-Cited by-同舟云学术

Human cytochromes P450 mediating phenacetin O‐deethylation in vitro: Validation of the high affinity component as an index of CYP1A2 activity

Published:1998-12 Issue:12 Volume:87 Page:1502-1507
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Venkatakrishnan Karthik,Moltke Lisa L.Von,Greenblatt David J.

Publisher

American Geophysical Union (AGU)

Subject

Pharmaceutical Science

Reference23 articles.

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3. Phenacetin O‐deethylation by human liver microsomes in vitro: inhibition by chemical probes, SSRI antidepres‐sants, nefazodone and venlafaxine;von Moltke;Psychopharmacology,1996

4. Furafylline is a potent and selective inhibitor of cytochrome P450 IA2 in man;Sesardic;Br. J. Clin. Pharmacol.,1990

5. Cytochrome P450 inhibitors: Evaluation of specificities in the in vitro metabolism of therapeutic agents by human liver microsomes;Newton;Drug Metab. Dispos.,1995

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