Efficient Asymmetric Synthesis of Novel Gastrin Receptor Antagonist AG-041R via Highly Stereoselective Alkylation of Oxindole Enolates-Reference-Cited by-同舟云学术

Efficient Asymmetric Synthesis of Novel Gastrin Receptor Antagonist AG-041R via Highly Stereoselective Alkylation of Oxindole Enolates

Published:2006-09-30 Issue:22 Volume:71 Page:8559-8564
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Emura Takashi¹,Esaki Toru¹,Tachibana Kazutaka¹,Shimizu Makoto¹

Affiliation:

1. Chemistry Research Department 1, Chugai Pharmaceutical Co., Ltd., 1-135 Komakado, Gotemba, Shizuoka 412-8513, Japan, and Department of Chemistry for Materials, Graduate School of Engineering, Mie University, 1577 Kurimamachiya-cho, Tsu, Mie 514-8507, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo061541v

Reference19 articles.

1. Pharmacological analysis of CCK2 receptor antagonists using isolated rat stomach ECL cells

2. Evaluation of Three Novel Cholecystokinin-B/Gastrin Receptor Antagonists: A Study of their Effects on Rat Stomach Enterochromaffin-Like Cell Activity

3. Stereoselective synthesis of quaternary α-amino acids. Part 1: Acyclic compounds

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