Structure−Activity Study on the Phe Side Chain Arrangement of Endomorphins Using Conformationally Constrained Analogues-Reference-Cited by-同舟云学术

Structure−Activity Study on the Phe Side Chain Arrangement of Endomorphins Using Conformationally Constrained Analogues

Published:2003-12-24 Issue:3 Volume:47 Page:735-743
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tömböly Csaba¹,Kövér Katalin E.¹,Péter Antal¹,Tourwé Dirk¹,Biyashev Dauren¹,Benyhe Sándor¹,Borsodi Anna¹,Al-Khrasani Mahmoud¹,Rónai András Z.¹,Tóth Géza¹

Affiliation:

1. Institute of Biochemistry, Biological Research Center of the Hungarian Academy of Sciences, 6701 Szeged, P.O. Box 521, Hungary; Department of Inorganic and Analytical Chemistry, University of Debrecen, 4010 Debrecen, P.O. Box 21, Hungary; Department of Inorganic and Analytical Chemistry, University of Szeged, 6701 Szeged, P.O. Box 440, Hungary; Department of Organic Chemistry, Vrije University Brussels, Pleinlaan 2, 1050 Brussels, Belgium; and Department of Pharmacology and Pharmacotherapy, Faculty of...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0310028

Reference63 articles.

1. A potent and selective endogenous agonist for the µ-opiate receptor

2. Localization of Endomorphin-2-Like Immunoreactivity in the Rat Medulla and Spinal Cord

3. Endomorphins fully activate a cloned human mu opioid receptor

4. The effects of endomorphin-1 and endomorphin-2 in CHO cells expressing recombinant μ-opioid receptors and SH-SY5Y cells

5. Activation and internalization of the μ-opioid receptor by the newly discovered endogenous agonists, endomorphin-1 and endomorphin-2

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