Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanylcarbamic Acid Esters, a Class of Potent N-Acylethanolamine Acid Amidase (NAAA) Inhibitors-Reference-Cited by-同舟云学术

Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanylcarbamic Acid Esters, a Class of Potent N-Acylethanolamine Acid Amidase (NAAA) Inhibitors

Published:2013-08-30 Issue:17 Volume:56 Page:6917-6934
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ponzano Stefano¹,Bertozzi Fabio¹,Mengatto Luisa¹,Dionisi Mauro¹,Armirotti Andrea¹,Romeo Elisa¹,Berteotti Anna¹,Fiorelli Claudio¹,Tarozzo Glauco¹,Reggiani Angelo¹,Duranti Andrea²,Tarzia Giorgio²,Mor Marco³,Cavalli Andrea¹⁴,Piomelli Daniele¹⁵,Bandiera Tiziano¹

Affiliation:

1. Drug Discovery and Development, Istituto Italiano di Tecnologia, Via Morego 30, I-16163 Genova, Italy

2. Dipartimento di Scienze Biomolecolari, Università degli Studi di Urbino “Carlo Bo”, Piazza del Rinascimento 6, I-61029 Urbino, Italy

3. Dipartimento di Farmacia, Università degli Studi di Parma, Viale delle Scienze 27/A, I-43124 Parma, Italy

4. Department of Pharmaceutical Sciences, University of Bologna, Via Belmeloro 6, I-40126, Bologna, Italy

5. Department of Anatomy and Neurobiology, Pharmacology and Biological Chemistry, University of California, Irvine, California 92697-4625, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400739u

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